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Cinnamic Acid Ameliorates Acetic Acid-induced Inflammatory Response through Inhibition of TLR-4 in Colitis Rat Model

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바이오화학분류
    • 바이오정밀화학
      1. 용매
    • 화장품용 기능성소재
      1. 계면활성제⁄증점제
    • 의료용 화학소재
      1. 식품첨가제
논문

Cinnamic Acid Ameliorates Acetic Acid-induced Inflammatory Response through Inhibition of TLR-4 in Colitis Rat Model

학술지

Anti-inflammatory & anti-allergy agents in medicinal chemistry

저자명

Rezaei, Zahra; Momtaz, Saeideh; Gharazi, Pardis; Rahimifard, Mahban; Baeeri, Maryam; Abdollahi, Ali Reza; Abdollahi, Mohammad; Niknejad, Amirhossein; Khayatan, Danial; Farzaei, Mohammad Hosein; Abdolghaffari, Amir Hossein

초록

<P>Background:<P>Cinnamic acid, an active compound in cinnamon spp., has anti-inflammatory and antioxidant characteristics and is favorable in managing inflammatory bowel diseases.</P></P><P>background:<P>Background: Cinnamic acid is a chemical with anti-inflammatory and antioxidant characteristics, thus might help to manage inflammatory bowel disease.</P></P><P>Objective:<P>Evaluate cinnamic acid's effects on colitis in rats.</P></P><P>Methods:<P>To induce colitis in experimental rats, excluding the sham group, a 4% intrarectal solu-tion of acetic acid was administered. The rats were then given oral doses of cinnamic acid at 30, 45, and 90 mg/kg for two days. The animals were assessed for macroscopic and microscopic changes, and the levels of inflammatory mediators such as tumor necrosis factor-alpha (TNF-&alpha;), interleukin-6 (IL-6), and myeloperoxidase (MPO) were measured using Eliza kits. Additionally, real-time PCR was performed to examine the gene level of toll-like receptor 4 (TLR-4) in the colon.</P></P><P>Results:<P>Effective reduction of inflammation in acetic acid-induced colitis was achieved through Cinnamic acid administration at doses of 45 and 90 mg/kg. The decrease was achieved by inhibiting the activities of TNF-&alpha;, IL-6, and MPO while downregulating the expression of TLR-4. It is important to note that macroscopic and microscopic evaluations were significant in determining the effectiveness of cinnamic acid in reducing inflammation.</P></P><P>Conclusion:<P>Downregulation of inflammatory cytokines and TLR-4 expression may contribute to cinnamic acid's anti-inflammatory effect.</P></P>

발행연도

2024

발행기관

Bentham Science

ISSN

1871-5230

23

페이지

pp.21-30

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1 2023-12-11

논문; 2024-01-01

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